Thiamine (Vitamin B1)

Brand Names: Benerva

Drug Class: Water-soluble vitamin (Vitamin B complex)

Overview

Thiamine (Vitamin B1) is an essential water-soluble vitamin that functions as a coenzyme in carbohydrate metabolism and energy production. It is used to treat and prevent thiamine deficiency, including conditions like beriberi and Wernicke-Korsakoff syndrome. Thiamine is generally well-tolerated with minimal toxicity.

Mechanism of Action

Thiamine acts as a coenzyme (thiamine pyrophosphate) in carbohydrate metabolism, facilitating decarboxylation of alpha-keto acids and transketolation in the pentose phosphate pathway. It is essential for energy production, nerve conduction, and myocardial function.

Indications

  • Treatment and prevention of thiamine deficiency (beriberi)
  • Wernicke-Korsakoff syndrome
  • Metabolic disorders requiring thiamine supplementation
  • Alcohol use disorder with nutritional deficiency

Common Doses

  • 50 mg tablet
  • 100 mg tablet
  • 100 mg/mL injection
  • 250 mg/mL injection

Dosage

Typical adult dosage for deficiency: 5-30 mg daily in divided doses; for severe deficiency (Wernicke's encephalopathy): 100 mg IV initially, then 50-100 mg IM/IV daily until clinical improvement. Maintenance: 5-10 mg daily orally.

Contraindications

  • Known hypersensitivity to thiamine or any component of the formulation

Side Effects

  • Generally well-tolerated
  • Rare hypersensitivity reactions (itching, urticaria, anaphylaxis)
  • Local irritation with parenteral administration
  • Nausea at high oral doses

Interactions

  • Loop diuretics (furosemide) may increase thiamine excretion
  • Chronic alcohol use impairs thiamine absorption and utilization

Counseling Points

  • Take with food to minimize gastrointestinal upset
  • Do not exceed recommended dosage without medical supervision
  • Store in a cool, dry place away from light and moisture
  • Inform healthcare provider if pregnant, planning pregnancy, or breastfeeding