Citicoline

Brand Names: Somazina

Drug Class: Psychostimulant; Nootropic agent

Overview

Citicoline is a brain chemical that occurs naturally in the body. As a medicine, it is used to treat stroke, head trauma, and age-related memory loss. It is also used for Parkinson's disease, glaucoma, and other conditions.

Mechanism of Action

Citicoline is a precursor of acetylcholine and phosphatidylcholine. It stabilizes cell membranes, reduces free radical formation, and increases neurotransmitter levels (acetylcholine, dopamine, norepinephrine). It also enhances brain metabolism and neuroprotection.

Indications

  • Stroke
  • Traumatic brain injury
  • Cognitive impairment in elderly
  • Parkinson's disease
  • Glaucoma

Dosage

Oral: 500-2000 mg daily in divided doses. For stroke: 500-2000 mg/day. For cognitive impairment: 500-1000 mg/day. Intravenous or intramuscular: 500-2000 mg/day. Use as directed by physician.

Contraindications

  • Hypersensitivity to citicoline or any component
  • Patients with severe renal impairment

Side Effects

  • Headache
  • Dizziness
  • Insomnia
  • Nausea
  • Diarrhea
  • Anorexia
  • Hypotension
  • Tachycardia
  • Allergic reactions

Interactions

  • Levodopa: may enhance effects
  • Anticholinergic drugs: may reduce effects
  • Other CNS stimulants: additive effects